Which of following statement about drug action is false ?
1) Competitive antagonist has no intrinsic activity but affinity
2) Competitive antagonist has intrinsic activity and affinity
3) Partial agonist has submaximal intrinsic activity and affinity
4) Inverse agonists have affinity but minus intrinsic activity.
๐ Explanation:
Competitive antagonists bind to receptors but do not activate them, meaning they have no intrinsic activity. They have affinity for the receptor, allowing them to compete with agonists for binding.